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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $34.85 | Total: $174.25 |
| 1 | 10 | $29.52 | Total: $295.20 |
| 1 | 25 | $25.01 | Total: $625.25 |
| 1 | 50 | $21.32 | Total: $1,066.00 |
| 1 | 100 | $18.45 | Total: $1,845.00 |
Overview
Vorasidenib (PVMMA) is an inhibitor of mutant isocitrate dehydrogenase (IDH; IC50s = 31.9 and 31.7 nM for IDH1R132H and IDH2R140Q, respectively)
Chemical Properties
| Molecular Formula | C14H13ClF6N6 |
| Molecular Weight | 414.74 |
| CAS Numbers | 1644545-52-7 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | C[C@@H](Nc1nc(N[C@H](C)C(F)(F)F)nc(n1)-c1cccc(Cl)n1)C(F)(F)F |
Storage and Handling
0C Short Term, -20C Long Term
References
Zakkula A, Dittakavi S, Maniyar MM,et al.Validated HPLC method for simultaneous quantification of mutant IDH12 inhibitors [enasidenib, ivosidenib and vorasidenib] in mouse plasma Application to a pharmacokinetic study[J].Biomed Chromatogr. 2019 Nov;33[11] e4658.