AZD-5672

AZD-5672

AT30260

CAS 780750-65-4

More details

1000 Items

$235.30

$235.30 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
15 $153.85 Total: $769.25
110 $130.32 Total: $1,303.20
125 $110.41 Total: $2,760.25
150 $94.12 Total: $4,706.00
1100 $81.45 Total: $8,145.00

Overview

AZD-5672 is an antagonist of CCR5 with an IC50 of 0.32 nM. AZD-5672 inhibits hERG cardiac ion channel binding and P-gp-mediated digoxin transport with IC50s of 7.3 ?M and 32 ?M. AZD-5672 can be used in studies about rheumatoid arthritis.

Chemical Properties

Molecular FormulaC32H38F2N2O5S2
Molecular Weight632.78
CAS Numbers780750-65-4
SolubilityDMSO
Purity98% by HPLC
SMILES CodeCCN(C1CCN(CC[C@H](c2ccc(cc2)S(C)(=O)=O)c2cc(F)cc(F)c2)CC1)C(=O)Cc1ccc(cc1)S(C)(=O)=O

Storage and Handling

0C Short Term, -20C Long Term

References

Elsby R, et al. The utility of in vitro data in making accurate predictions of human P-glycoprotein-mediated drug-drug interactions a case study for AZD5672. Drug Metab Dispos. 2011 Feb;39[2] 275-82.