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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $31.45 | Total: $157.25 |
| 1 | 10 | $26.64 | Total: $266.40 |
| 1 | 25 | $22.57 | Total: $564.25 |
| 1 | 50 | $19.24 | Total: $962.00 |
| 1 | 100 | $16.65 | Total: $1,665.00 |
Overview
Ro 31-8220 Mesylate (Bisindolylmaleimide IX mesylate) is a pan-PKC inhibitor for PKC-??I?II?? (IC50: 524142724 nM), and also shows potent inhibition against MSK1, MAPKAP-K1b, S6K1, and GSK3?.
Chemical Properties
| Molecular Formula | C25H23N5O2S |
| Molecular Weight | 553.65 |
| CAS Numbers | 138489-18-6 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CS(O)(=O)=O.Cn1cc(C2=C(C(=O)NC2=O)c2cn(CCCSC(N)=N)c3ccccc23)c2ccccc12 |
Storage and Handling
0C Short Term, -20C Long Term
References
Wilkinson SE, et al. Biochem J. 1993, 294 [ Pt 2], 335-337.