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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $152.15 | Total: $760.75 |
| 1 | 10 | $128.88 | Total: $1,288.80 |
| 1 | 25 | $109.19 | Total: $2,729.75 |
| 1 | 50 | $93.08 | Total: $4,654.00 |
| 1 | 100 | $80.55 | Total: $8,055.00 |
Overview
Teglarinad chloride (GMX-1777 chloride) is a potent inhibitor of NAMPT, the precursor of GMX1778.Teglarinad chloride has antitumor activity and acts by interfering with DNA repair and inhibiting angiogenesis.
Chemical Properties
| Molecular Formula | C30H43Cl2N5O8 |
| Molecular Weight | 672.6 |
| CAS Numbers | 432037-57-5 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | [Cl-].COCCOCCOCCOCCOC(=O)OC[n+]1ccc(NC(NC#N)=NCCCCCCOc2ccc(Cl)cc2)cc1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Beauparlant P, et, al. Preclinical development of the nicotinamide phosphoribosyl transferase inhibitor prodrug GMX1777. Anticancer Drugs. 2009 Jun;20[5] 346-54.