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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $27.20 | Total: $136.00 |
| 1 | 10 | $23.04 | Total: $230.40 |
| 1 | 25 | $19.52 | Total: $488.00 |
| 1 | 50 | $16.64 | Total: $832.00 |
| 1 | 100 | $14.40 | Total: $1,440.00 |
Overview
Maritoclax (Marinopyrrole A) (Marinopyrrole A) is a novel and specific Mcl-1 inhibitor, shows >8 fold selectivity than BCL-xl (IC50 > 80 ?M),with an IC50 value of 10.1 ?M.
Chemical Properties
| Molecular Formula | C22H12Cl4N2O4 |
| Molecular Weight | 510.15 |
| CAS Numbers | 1227962-62-0 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Oc1ccccc1C(=O)c1[nH]c(Cl)c(Cl)c1-n1c(Cl)c(Cl)cc1C(=O)c1ccccc1O |
Storage and Handling
0C Short Term, -20C Long Term
References
Doi K, et al. Discovery of marinopyrrole A [maritoclax] as a selective Mcl-1 antagonist that overcomes ABT-737 resistance by binding to and targeting Mcl-1 for proteasomal degradation. J Biol Chem. 2012 Mar 23;287[13] 10224-35.