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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $602.65 | Total: $3,013.25 |
| 1 | 10 | $510.48 | Total: $5,104.80 |
| 1 | 25 | $432.49 | Total: $10,812.26 |
| 1 | 50 | $368.68 | Total: $18,434.00 |
| 1 | 100 | $319.05 | Total: $31,905.01 |
Overview
Ecopladib (PLA 725) is a sub-micromolar inhibitor of cytosolic phospholipase A2? (cPLA2?), with IC50s of 0.15 ?M and 0.11 ?M in the GLU micelle and rat whole blood assays, respectively.
Chemical Properties
| Molecular Formula | C39H33Cl3N2O5S |
| Molecular Weight | 748.11 |
| CAS Numbers | 381683-92-7 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | OC(=O)c1ccc(OCCc2c(CCNS(=O)(=O)Cc3ccc(Cl)c(Cl)c3)n(C(c3ccccc3)c3ccccc3)c3ccc(Cl)cc23)cc1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Lee KL, et al. Discovery of Ecopladib, an indole inhibitor of cytosolic phospholipase A2alpha. J Med Chem. 2007 Mar 22;50[6] 1380-400. Epub 2007 Feb 17.