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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $60.35 | Total: $301.75 |
| 1 | 10 | $51.12 | Total: $511.20 |
| 1 | 25 | $43.31 | Total: $1,082.75 |
| 1 | 50 | $36.92 | Total: $1,846.00 |
| 1 | 100 | $31.95 | Total: $3,195.00 |
Overview
TG 100801 is a dual inhibitor of VEGFr2 and Src family (Src and YES) kinases and is a candidate compound for the treatment of age-related macular degeneration (AMD).
Chemical Properties
| Molecular Formula | C33H30ClN5O3 |
| Molecular Weight | 580.08 |
| CAS Numbers | 867331-82-6 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cc1cc(cc2nnc(Nc3ccc(OCCN4CCCC4)cc3)nc12)-c1cc(OC(=O)c2ccccc2)ccc1Cl |
Storage and Handling
0C Short Term, -20C Long Term
References
Palanki MS, et al. Development of prodrug 4-chloro-3-[5-methyl-3-{[4-[2-pyrrolidin-1-ylethoxy]phenyl]amino}-1,2,4-benzotriazin-7-yl]phenyl benzoate [TG100801] a topically administered therapeutic candidate in clinical trials for the treatment of age-related macular degeneration. J Med Chem. 2008 Mar 27;51[6] 1546-59.