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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $59.50 | Total: $297.50 |
| 1 | 10 | $50.40 | Total: $504.00 |
| 1 | 25 | $42.70 | Total: $1,067.50 |
| 1 | 50 | $36.40 | Total: $1,820.00 |
| 1 | 100 | $31.50 | Total: $3,150.00 |
Overview
MLS000544460 is a highly selective and reversible Eya2 phosphatase inhibitor (Kd: 2.0 ?M, IC50: 4 ?M) that exhibits inhibitory effects on Eya2 phosphatase-mediated cell migration and has anticancer activity.
Chemical Properties
| Molecular Formula | C17H12FN3O2S |
| Molecular Weight | 341.36 |
| CAS Numbers | 352336-36-8 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Fc1cccc(c1)C(=O)NN=Cc1ccc(Sc2ccccn2)o1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Krueger AB, et al. Allosteric inhibitors of the Eya2 phosphatase are selective and inhibit Eya2-mediated cellmigration. J Biol Chem. 2014 Jun 6;289[23] 16349-61.