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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $31.45 | Total: $157.25 |
| 1 | 10 | $26.64 | Total: $266.40 |
| 1 | 25 | $22.57 | Total: $564.25 |
| 1 | 50 | $19.24 | Total: $962.00 |
| 1 | 100 | $16.65 | Total: $1,665.00 |
Overview
CCG-63808 is a reversible inhibitor of regulator of G-protein signaling (RGS) proteins, dose-dependently inhibiting the TR-FRET signal between RGS4-AF488 and Tb-G?o with an IC50 value of 1.9 ?M.
Chemical Properties
| Molecular Formula | C25H15FN4O2S |
| Molecular Weight | 454.48 |
| CAS Numbers | 620113-73-7 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cc1cccn2c1nc(Oc1ccc(F)cc1)c(C=C(C#N)c1nc3ccccc3s1)c2=O |
Storage and Handling
0C Short Term, -20C Long Term
References
Levi L. Blazer et al.Reversible, Allosteric Small-Molecule Inhibitors of Regulator of G Protein Signaling Proteins. Molecular Pharmacology September 2010 vol.78 no.3 524-533