Categories
- PROTAC Linker
- Protein Control Ligand
- Pathway Inhibitors
- Function Modulators
- Activators
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- Nuclear Receptor Ligands
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- TNF Receptors
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $24.65 | Total: $123.25 |
| 1 | 10 | $20.88 | Total: $208.80 |
| 1 | 25 | $17.69 | Total: $442.25 |
| 1 | 50 | $15.08 | Total: $754.00 |
| 1 | 100 | $13.05 | Total: $1,305.00 |
Overview
AS1517499 is a potent STAT6 inhibitor with IC50 of 21 nM
Chemical Properties
| Molecular Formula | C20H20ClN5O2 |
| Molecular Weight | 397.86 |
| CAS Numbers | 919486-40-1 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | NC(=O)c1cnc(NCCc2ccc(O)c(Cl)c2)nc1NCc1ccccc1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Nagashima S, et al. Synthesis and evaluation of 2-{[2-[4-hydroxyphenyl]-ethyl]amino}pyrimidine-5-carboxamide derivatives as novel STAT6 inhibitors. Bioorg Med Chem. 2007 Jan 15;15[2] 1044-55.