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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $29.75 | Total: $148.75 |
| 1 | 10 | $25.20 | Total: $252.00 |
| 1 | 25 | $21.35 | Total: $533.75 |
| 1 | 50 | $18.20 | Total: $910.00 |
| 1 | 100 | $15.75 | Total: $1,575.00 |
Overview
ALOX15-IN-2 is a potent inhibitor of ALOX15 linoleate oxygenase activity, inhibiting the oxidation of linoleic acid (LA) and arachidonic acid (AA), the immediate homologs of ALOX15, with IC50s of 1.55 and 2.79 ?M, respectively.
Chemical Properties
| Molecular Formula | C23H29N3O4S |
| Molecular Weight | 443.56 |
| CAS Numbers | 2764818-23-5 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | N(S(NC(OCCCCCCCC)=O)(=O)=O)C=1C=C(C2=CC=3C(N2)=CC=CC3)C=CC1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Golovanov A, et al. N-Substituted 5-[1H-Indol-2-yl]-2-methoxyanilines Are Allosteric Inhibitors of the Linoleate Oxygenase Activity of Selected Mammalian ALOX15 Orthologs Mechanism of Action. J Med Chem. 2022;65[3] 1979-1995.