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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $24.65 | Total: $123.25 |
| 1 | 10 | $20.88 | Total: $208.80 |
| 1 | 25 | $17.69 | Total: $442.25 |
| 1 | 50 | $15.08 | Total: $754.00 |
| 1 | 100 | $13.05 | Total: $1,305.00 |
Overview
CVT-12012 is an orally bioavailable inhibitor of stearoyl-CoA desaturase (SCD; IC50 = 6.1 nM in HepG2 cells).
Chemical Properties
| Molecular Formula | C21H21F3N4O3 |
| Molecular Weight | 434.41 |
| CAS Numbers | 1018675-35-8 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cc1nc2ccc(NCc3cccc(c3)C(F)(F)F)cc2n(CCNC(=O)CO)c1=O |
Storage and Handling
0C Short Term, -20C Long Term
References
Koltun D O , Vasilevich N I , Parkhill E Q , et al. Orally bioavailable, liver-selective stearoyl-CoA desaturase [SCD] inhibitors[J]. Bioorganic and Medicinal Chemistry Letters, 2009, 19[11] 3050-3053.