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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $158.10 | Total: $790.50 |
| 1 | 10 | $133.92 | Total: $1,339.20 |
| 1 | 25 | $113.46 | Total: $2,836.50 |
| 1 | 50 | $96.72 | Total: $4,836.00 |
| 1 | 100 | $83.70 | Total: $8,370.00 |
Overview
Stafib-2 is a potent and selective inhibitor of the transcription factor STAT5b, with IC50 values of 82 nM and 1.7 ?M for STAT5b and STAT5a, respectively. Stafib-2 has poor cell permeability.
Chemical Properties
| Molecular Formula | C28H26N2O12P2 |
| Molecular Weight | 644.46 |
| CAS Numbers | 2097938-74-2 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | O(P(=O)(O)O)C1=C(OP(=O)(O)O)C=CC(CNC(COC2=CC=C(C(NC3=CC=C(OC4=CC=CC=C4)C=C3)=O)C=C2)=O)=C1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Elumalai N, et al. Rational development of Stafib-2 a selective, nanomolar inhibitor of the transcription factor STAT5b. Sci Rep. 2017;7[1] 819.