ELA-11 (human) acetate(1784687-32-6 free base)

ELA-11 (human) acetate(1784687-32-6 free base)

ATP1922L1

1000 Items

$146.90

$146.90 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
15 $96.05 Total: $480.25
110 $81.36 Total: $813.60
125 $68.93 Total: $1,723.25
150 $58.76 Total: $2,938.00
1100 $50.85 Total: $5,085.00

Overview

ELA-11 (human) acetate high affinity apelin receptor agonist (Ki = 14 nM). Bioactive fragment of ELA-32. Inhibits forskolin-induced cAMP production and stimulates ?-arrestin recruitment in vitro.

Chemical Properties

Molecular FormulaC60H94N16O15S2
Molecular Weight1343.61
SolubilityDMSO
Purity98% by HPLC
SMILES CodeO=C(N1[C@@H](CCC1)C(O)=O)[C@H](CC2=CC=CC=C2)NC([C@H]3N(CCC3)C([C@H](C(C)C)NC([C@H](CCCNC(N)=N)NC([C@H](CO)NC([C@@H](NC([C@H](CC(C)C)NC([C@H]4N(CCC4)C([C@H](CCSC)NC([C@@H](N)CS)=O)=O)=O)=O)CC5=CN=CN5)=O)=O)=O)=O)=O.CC(O)=O

Storage and Handling

0C Short Term, -20C Long Term

References

Yang et al [2017] ElabelaToddler is an endogenous agonist of the apelin APJ receptor in the adult cardiovascular system, and exogenous administration of the peptide compensates for the downregulation of its expression in pulmonary arterial hypertension. Circulation 135 1160 PMID