Categories
- PROTAC Linker
- Protein Control Ligand
- Pathway Inhibitors
- Function Modulators
- Activators
- G Protein-Coupled Receptor Ligands
- Nuclear Receptor Ligands
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- TNF Receptors
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $84.15 | Total: $420.75 |
| 1 | 10 | $71.28 | Total: $712.80 |
| 1 | 25 | $60.39 | Total: $1,509.75 |
| 1 | 50 | $51.48 | Total: $2,574.00 |
| 1 | 100 | $44.55 | Total: $4,455.00 |
Overview
NEO2734 (EP31670) is an orally active, selective inhibitor of p300CBP and BET bromodomains, with an IC50 of less than 30 nM for both targets.
Chemical Properties
| Molecular Formula | C22H24F3N3O3 |
| Molecular Weight | 435.44 |
| CAS Numbers | 2081072-29-7 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cc1cc(cn(C)c1=O)-c1ccc2nc(C3CCOCC3)n(CCOC(F)(F)F)c2c1 |
Storage and Handling
0C Short Term, -20C Long Term
References
The novel BET-CBPp300 dual inhibitor NEO2734 is active in SPOP mutant and wild-type prostate cancer