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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $61.20 | Total: $306.00 |
| 1 | 10 | $51.84 | Total: $518.40 |
| 1 | 25 | $43.92 | Total: $1,098.00 |
| 1 | 50 | $37.44 | Total: $1,872.00 |
| 1 | 100 | $32.40 | Total: $3,240.00 |
Overview
CPI-1205 is a highly potent and selective inhibitor of EZH2(IC50 : 0.002 ?M, EC50 : 0.032 ?M) .
Chemical Properties
| Molecular Formula | C27H33F3N4O3 |
| Molecular Weight | 518.57 |
| CAS Numbers | 1621862-70-1 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | [C@H](C)(N1C=2C(C(C(NCC3=C(OC)C=C(C)NC3=O)=O)=C1C)=CC=CC2)C4CCN(CC(F)(F)F)CC4 |
Storage and Handling
0C Short Term, -20C Long Term
References
Vaswani RG, et al. Identification of [R]-N-[[4-Methoxy-6-methyl-2-oxo-1,2-dihydropyridin-3-yl]methyl]-2-methyl-1-[1-[1-[2,2,2-trifluoroethyl]piperidin-4-yl]ethyl]-1H-indole-3-carboxamide [CPI-1205], a Potent and Selective Inhibitor of Histone Methyltransferase EZH2, Suitable for Phase I Clinical Trials for B-Cell Lymphomas. J Med Chem. 2016 Nov 10;59[21] 9928-9941.