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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $211.65 | Total: $1,058.25 |
| 1 | 10 | $179.28 | Total: $1,792.80 |
| 1 | 25 | $151.89 | Total: $3,797.25 |
| 1 | 50 | $129.48 | Total: $6,474.00 |
| 1 | 100 | $112.05 | Total: $11,205.00 |
Overview
MIV-6R inhibits Menin-MLL interaction (IC50: 56 nM) and can be used to study leukemia.
Chemical Properties
| Molecular Formula | C27H35N3O |
| Molecular Weight | 417.59 |
| CAS Numbers | 1560968-55-9 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | [C@@](N)([C@@H]1CCN(CCCOC2=CC=C(C#N)C=C2)CC1)(C3CCCC3)C4=CC=CC=C4 |
Storage and Handling
0C Short Term, -20C Long Term
References
He S, Senter TJ, Pollock J, Han C, Upadhyay SK, Purohit T, Gogliotti RD, Lindsley CW, Cierpicki T, Stauffer SR, Grembecka J. High-affinity small-molecule inhibitors of the menin-mixed lineage leukemia [MLL] interaction closely mimic a natural protein-protein interaction. J Med Chem. 2014 Feb 27;57[4] 1543-56. doi 10.1021jm401868d. Epub 2014 Feb 6. PubMed PMID 24472025; PubMed Central PMCID PMC3983337.