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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $129.20 | Total: $646.00 |
| 1 | 10 | $109.44 | Total: $1,094.40 |
| 1 | 25 | $92.72 | Total: $2,318.00 |
| 1 | 50 | $79.04 | Total: $3,952.00 |
| 1 | 100 | $68.40 | Total: $6,840.00 |
Overview
Vafidemstat (ORY-2001) is a selective, orally active lysyl-histone demethylase (LSD1)MAO-B inhibitor that crosses the blood-brain barrier for the study of neurological diseases.
Chemical Properties
| Molecular Formula | C19H20N4O2 |
| Molecular Weight | 336.39 |
| CAS Numbers | 1357362-02-7 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Nc1nnc(CN[C@@H]2C[C@H]2c2ccc(OCc3ccccc3)cc2)o1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Antonijoan RM,et al. First-in-Human Randomized Trial to Assess Safety, Tolerability, Pharmacokinetics and Pharmacodynamics of the KDM1A Inhibitor Vafidemstat. CNS Drugs. 2021 Mar;35[3] 331-344.