Categories
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $70.55 | Total: $352.75 |
| 1 | 10 | $59.76 | Total: $597.60 |
| 1 | 25 | $50.63 | Total: $1,265.75 |
| 1 | 50 | $43.16 | Total: $2,158.00 |
| 1 | 100 | $37.35 | Total: $3,735.00 |
Overview
OTS186935 FA is a protein methyltransferase SUV39H2 inhibitor.OTS186935 FA inhibits tumor growth in MDA-MB-231 breast cancer cells and A549 lung cancer cells.
Chemical Properties
| Molecular Formula | C26H28ClN5O4 |
| Molecular Weight | 509.98 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | COC1=C(C2=CN(C=CC(N3C[C@H](CC3)NCC4=CC=NC=C4)=C5)C5=N2)C=C(C(OC)=C1)Cl.[H]C(O)=O |
Storage and Handling
0C Short Term, -20C Long Term
References
Vougiouklakis T, et al. Development of novel SUV39H2 inhibitors that exhibit growth suppressive effects in mouse xenograft models and regulate the phosphorylation of H2AX. Oncotarget. 2018 Aug 7;9[61] 31820-31831.