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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $567.80 | Total: $2,839.00 |
| 1 | 10 | $480.96 | Total: $4,809.60 |
| 1 | 25 | $407.48 | Total: $10,187.01 |
| 1 | 50 | $347.36 | Total: $17,368.00 |
| 1 | 100 | $300.60 | Total: $30,060.01 |
Overview
T-448 is a specific, orally active, and irreversible inhibitor of lysine-specific demethylase 1 (LSD1, an H3K4 demethylase) with an IC50 of 22 nM.
Chemical Properties
| Molecular Formula | C19H22N4O3S |
| Molecular Weight | 386.47 |
| CAS Numbers | 1597426-53-3 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | C(=CC(O)=O)C(O)=O.N([C@H]1[C@@H](C1)C2=CC(C(NC3=NN=C(C)S3)=O)=CC=C2)C4CCC4 |
Storage and Handling
0C Short Term, -20C Long Term
References
Matsuda S, et al. T-448, a specific inhibitor of LSD1 enzyme activity, improves learning function without causing thrombocytopenia in mice. Neuropsychopharmacology. 2018 Dec 22.