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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $41.65 | Total: $208.25 |
| 1 | 10 | $35.28 | Total: $352.80 |
| 1 | 25 | $29.89 | Total: $747.25 |
| 1 | 50 | $25.48 | Total: $1,274.00 |
| 1 | 100 | $22.05 | Total: $2,205.00 |
Overview
ZEN-3862 (Willardiine) is an inhibitor of BET(IC50s of 0.16 and 0.13 ?M for BRD4(BD1) and BRD4(BD2) , respectively). ZEN-3862 can be used to form PROTACs to induce degradation of BRD4.
Chemical Properties
| Molecular Formula | C19H17FN2O3 |
| Molecular Weight | 340.35 |
| CAS Numbers | 1952264-33-3 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CC=1C(C2=CN(CC3=CC(F)=C(C=C3)C4CO4)C(=O)C=C2)=C(C)ON1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Kharenko OA, et al. Design and Characterization of Novel Covalent Bromodomain and Extra-Terminal Domain [BET] Inhibitors Targeting a Methionine. J Med Chem. 2018 Sep 27;61[18] 8202-8211.