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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $327.25 | Total: $1,636.25 |
| 1 | 10 | $277.20 | Total: $2,772.00 |
| 1 | 25 | $234.85 | Total: $5,871.25 |
| 1 | 50 | $200.20 | Total: $10,010.00 |
| 1 | 100 | $173.25 | Total: $17,325.01 |
Overview
C-82 is a specific CBP?-catenin antagonist. It inhibits the binding between ?-catenin and CBP and increases the binding between ?-catenin and p300.
Chemical Properties
| Molecular Formula | C33H34N6O4 |
| Molecular Weight | 578.66 |
| CAS Numbers | 1422253-37-9 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | [H][C@]12[C@H](C)N(Cc3cccc4cccnc34)C(=O)[C@H](Cc3ccc(O)cc3)N1C(=O)CN(C)N2C(=O)NCc1ccccc1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Osawa Y, et al. Inhibition of Cyclic Adenosine Monophosphate [cAMP]-response Element-binding Protein [CREB]-binding Protein [CBP]?-Catenin Reduces Liver Fibrosis in Mice. EBioMedicine. 2015 Oct 8;2[11] 1751-8.