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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $69.70 | Total: $348.50 |
| 1 | 10 | $59.04 | Total: $590.40 |
| 1 | 25 | $50.02 | Total: $1,250.50 |
| 1 | 50 | $42.64 | Total: $2,132.00 |
| 1 | 100 | $36.90 | Total: $3,690.00 |
Overview
OXFBD04 is a potent and selective BRD4 inhibitor (IC50= 166 nM), a BET bromodomain ligand with modest affinity for the CREBBP bromodomain, and exhibits anti-cancer activity.
Chemical Properties
| Molecular Formula | C17H16N2O3 |
| Molecular Weight | 296.32 |
| CAS Numbers | 2231747-03-6 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cc1noc(C)c1-c1cc(O)cc(c1)C(O)c1cccnc1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Jennings LE, et al. BET bromodomain ligands Probing the WPF shelf to improve BRD4 bromodomain affinity and metabolic stability. Bioorg Med Chem. 2018 Jul 15;26[11] 2937-2957.