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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $29.75 | Total: $148.75 |
| 1 | 10 | $25.20 | Total: $252.00 |
| 1 | 25 | $21.35 | Total: $533.75 |
| 1 | 50 | $18.20 | Total: $910.00 |
| 1 | 100 | $15.75 | Total: $1,575.00 |
Overview
BVT948 is a protein tyrosine phosphatase (PTP) inhibitor that also inhibits lysine methyltransferase SETD8 (KMT5A) and various cytochrome P450 (P450) isoforms.
Chemical Properties
| Molecular Formula | C14H11NO3 |
| Molecular Weight | 241.24 |
| CAS Numbers | 39674-97-0 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CC1(C)C(=O)N=C2C1=C(O)C(=O)c1ccccc21 |
Storage and Handling
0C Short Term, -20C Long Term
References
Liljebris C, et al. Oxidation of protein tyrosine phosphatases as a pharmaceutical mechanism of action a study using 4-hydroxy-3,3-dimethyl-2H-benzo[g]indole-2,5[3H]-dione. J Pharmacol Exp Ther. 2004 May;309[2] 711-9.