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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $200.60 | Total: $1,003.00 |
| 1 | 10 | $169.92 | Total: $1,699.20 |
| 1 | 25 | $143.96 | Total: $3,599.00 |
| 1 | 50 | $122.72 | Total: $6,136.00 |
| 1 | 100 | $106.20 | Total: $10,620.00 |
Overview
MPI_5a is an effective and selective inhibitor of HDAC6 (IC50=36 nM). MPI_5a weakly inhibits other HDAC isoforms and it also inhibits acyl-tubulin accumulation in cells (IC50: 210 nM).
Chemical Properties
| Molecular Formula | C16H17N3O3 |
| Molecular Weight | 299.32 |
| CAS Numbers | 1259296-46-2 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | C(=O)(N1CC=2C(=CC(C(NO)=O)=CC2)CC1)C=3N(C)C=CC3 |
Storage and Handling
0C Short Term, -20C Long Term
References
Blackburn C, et al. Potent histone deacetylase inhibitors derived from 4-[aminomethyl]-N-hydroxybenzamide with high selectivity for the HDAC6 isoform. J Med Chem. 2013 Sep 26;56[18] 7201-11.