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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $53.55 | Total: $267.75 |
| 1 | 10 | $45.36 | Total: $453.60 |
| 1 | 25 | $38.43 | Total: $960.75 |
| 1 | 50 | $32.76 | Total: $1,638.00 |
| 1 | 100 | $28.35 | Total: $2,835.00 |
Overview
GSK467 is a potent and selective inhibitor of KDM5 (JARID1)(Ki : 10 nM).
Chemical Properties
| Molecular Formula | C17H13N5O2 |
| Molecular Weight | 319.32 |
| CAS Numbers | 1628332-52-4 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | O=c1[nH]c(Oc2cnn(Cc3ccccc3)c2)nc2cnccc12 |
Storage and Handling
0C Short Term, -20C Long Term
References
Johansson C, et al. Structural analysis of human KDM5B guides histone demethylase inhibitor development. Nat Chem Biol. 2016 Jul;12[7] 539-45.