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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $39.95 | Total: $199.75 |
| 1 | 10 | $33.84 | Total: $338.40 |
| 1 | 25 | $28.67 | Total: $716.75 |
| 1 | 50 | $24.44 | Total: $1,222.00 |
| 1 | 100 | $21.15 | Total: $2,115.00 |
Overview
ZEN-2759 is a potent BET small molecule inhibitor of BRD4 (BD1), BRD4 (BD2), and BRD4 (BD1BD2).
Chemical Properties
| Molecular Formula | C17H16N2O2 |
| Molecular Weight | 280.32 |
| CAS Numbers | 1616400-50-0 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CC=1C(C2=CN(CC3=CC=CC=C3)C(=O)C=C2)=C(C)ON1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Kharenko OA, et al. Design and Characterization of Novel Covalent Bromodomain and Extra-Terminal Domain [BET] Inhibitors Targeting a Methionine. J Med Chem. 2018 Sep 27;61[18] 8202-8211.