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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $37.40 | Total: $187.00 |
| 1 | 10 | $31.68 | Total: $316.80 |
| 1 | 25 | $26.84 | Total: $671.00 |
| 1 | 50 | $22.88 | Total: $1,144.00 |
| 1 | 100 | $19.80 | Total: $1,980.00 |
Overview
BAY 598 is a potent and selective competitive inhibitor of SMYD2 lysine methyltransferase, IC50 values are 27 and 58 nM for biochemical and cellular activity assays, respectively.
Chemical Properties
| Molecular Formula | C22H20Cl2F2N6O3 |
| Molecular Weight | 525.34 |
| CAS Numbers | 1906919-67-2 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CCN([C@H]1CN(N=C1c1ccc(Cl)c(Cl)c1)C(NC#N)=Nc1cccc(OC(F)F)c1)C(=O)CO |
Storage and Handling
0C Short Term, -20C Long Term
References
Reynoird N , Mazur P K , Stellfeld T , et al. Coordination of stress signals by the lysine methyltransferase SMYD2 promotes pancreatic cancer[J]. Genes & Development, 2016 genesdev;gad.275529.115v1.