Categories
- PROTAC Linker
- Protein Control Ligand
- Pathway Inhibitors
- Function Modulators
- Activators
- G Protein-Coupled Receptor Ligands
- Nuclear Receptor Ligands
- GDNF Receptors
- TNF Receptors
- Transcription Factors
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- Customized Screening Library
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- Primary Cells
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $85.00 | Total: $425.00 |
| 1 | 10 | $72.00 | Total: $720.00 |
| 1 | 25 | $61.00 | Total: $1,525.00 |
| 1 | 50 | $52.00 | Total: $2,600.00 |
| 1 | 100 | $45.00 | Total: $4,500.00 |
Overview
JG-2016, as a small molecule histone acetyltransferase 1 (HAT1) inhibitor, inhibits the growth of human cancer cell lines, inhibits enzyme activity in cellulose, and interferes with tumor growth.
Chemical Properties
| Molecular Formula | C18H21ClN4O3 |
| Molecular Weight | 376.84 |
| CAS Numbers | 2887480-87-5 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | O=C1N=C2C(=NC=3C=C(Cl)C(=CC3N2CCOCC(C)C)CC)C(=O)N1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Gaddameedi JD,et al. Acetyl-Click Screening Platform Identifies Small-Molecule Inhibitors of Histone Acetyltransferase 1 [HAT1]. J Med Chem. 2023 Apr 27;66[8] 5774-5801.