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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $28.05 | Total: $140.25 |
| 1 | 10 | $23.76 | Total: $237.60 |
| 1 | 25 | $20.13 | Total: $503.25 |
| 1 | 50 | $17.16 | Total: $858.00 |
| 1 | 100 | $14.85 | Total: $1,485.00 |
Overview
SGC-SMARCA-BRDVIII is a potent and selective inhibitor of SMARCA2, SMARCA4, PB1(2), PB1(3), and PB1(5) with Kds of 35 nM, 36 nM, 3.7 ?M, 2.0 ?M, and 13 nM, respectively.
Chemical Properties
| Molecular Formula | C19H25N5O3 |
| Molecular Weight | 371.43 |
| CAS Numbers | 1997319-84-2 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CC(C)(C)OC(=O)N1CCN(CC1)c1cc(nnc1N)-c1ccccc1O |
Storage and Handling
0C Short Term, -20C Long Term
References
Wanior M, et, al. Pan-SMARCAPB1 Bromodomain Inhibitors and Their Role in Regulating Adipogenesis. J Med Chem. 2020 Dec 10;63[23] 14680-14699.