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Overview
Rupatadine Fumarate (Rinialer) (UR-12592 Fumarate) is a potent dual PAFH1 antagonist with Ki of 0.550.1 uM.
Chemical Properties
| Molecular Formula | C26H26ClN3 |
| Molecular Weight | 532.03 |
| CAS Numbers | 182349-12-8 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | OC(=O)C=CC(O)=O.Cc1cncc(CN2CCC(CC2)=C2c3ccc(Cl)cc3CCc3cccnc23)c1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Merlos M, et al. J Pharmacol Exp Ther, 1997, 280[1], 114-121.