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![d[Leu4,Lys8]-VP acetate](https://img.aobious.com/img/p/4/9/5/4/9/49549-large_default.webp "d[Leu4,Lys8]-VP acetate")
![d[Leu4,Lys8]-VP acetate](https://img.aobious.com/img/p/4/9/5/4/9/49549.jpg "d[Leu4,Lys8]-VP acetate")
Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $28.05 | Total: $140.25 |
| 1 | 10 | $23.76 | Total: $237.60 |
| 1 | 25 | $20.13 | Total: $503.25 |
| 1 | 50 | $17.16 | Total: $858.00 |
| 1 | 100 | $14.85 | Total: $1,485.00 |
Overview
d[Leu4,Lys8]-VP acetate is a selective vasopressin V1b receptor agonist. The Kis for rat, human and mouse V1b receptors are 0.16 nM, 0.52 nM and 0.1.38 nM, respectively. d[Leu4,Lys8]-VP acetate exhibits weak antidiuretic, vasopressor and oxytocic activiti
Chemical Properties
| Molecular Formula | C49H71N11O13S2 |
| Molecular Weight | 1086.28 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CC(O)=O.NC(CNC([C@@H](NC([C@@H]1CCCN1C([C@@H](NC([C@@H]2CC(N)=O)=O)CSSCCC(N[C@H](C(N[C@](CC3=CC=CC=C3)([H])C(N[C@@H](CC(C)C)C(N2)=O)=O)=O)CC4=CC=C(O)C=C4)=O)=O)=O)CCCCN)=O)=O |
Storage and Handling
0C Short Term, -20C Long Term
References
Ana P, et, al. Design and synthesis of the first selective agonists for the rat vasopressin V[1b] receptor based on modifications of deamino-[Cys1]arginine vasopressin at positions 4 and 8. J Med Chem. 2007 Feb 22; 50[4] 835-47.