Categories
- PROTAC Linker
- Protein Control Ligand
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $95.20 | Total: $476.00 |
| 1 | 10 | $80.64 | Total: $806.40 |
| 1 | 25 | $68.32 | Total: $1,708.00 |
| 1 | 50 | $58.24 | Total: $2,912.00 |
| 1 | 100 | $50.40 | Total: $5,040.00 |
Overview
E7016 (GPI 21016) is an orally available PARP inhibitor that inhibits DNA repair and enhances tumor cell radiosensitivity both in vitro and in vivo.
Chemical Properties
| Molecular Formula | C20H19N3O3 |
| Molecular Weight | 349.38 |
| CAS Numbers | 902128-92-1 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | OC1CCN(Cc2ccc3oc4cccc5c4c(n[nH]c5=O)c3c2)CC1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Andrea L Russo, et al. In vitro and in vivo radiosensitization of glioblastoma cells by the poly [ADP-ribose] polymerase inhibitor E7016. Clin Cancer Res. 2009 Jan 15;15[2] 607-12.