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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $64.60 | Total: $323.00 |
| 1 | 10 | $54.72 | Total: $547.20 |
| 1 | 25 | $46.36 | Total: $1,159.00 |
| 1 | 50 | $39.52 | Total: $1,976.00 |
| 1 | 100 | $34.20 | Total: $3,420.00 |
Overview
SHU 9119 acetate is a well-known antagonist of human melanocortin 3 and 4 (hMC3R, hMC4R) receptors and a partial hMC5R agonist. The IC50 values of human MC3R, MC4R and MC5R is 0.23, 0.06, and 0.09 nM respectively.
Chemical Properties
| Molecular Formula | C56H75N15O11 |
| Molecular Weight | 1134.29 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CCCC[C@@H](C(N[C@H]1CC(NCCCC[C@@H](C(N)=O)NC([C@@H](NC([C@@H](NC([C@H](NC([C@@H](NC1=O)CC2=CNC=N2)=O)CC3=CC4=CC=CC=C4C=C3)=O)CCCNC(N)=N)=O)CC5=CNC6=C5C=CC=C6)=O)=O)=O)NC(C)=O.CC(O)=O |
Storage and Handling
0C Short Term, -20C Long Term
References
Grieco P, et al. Further structure-activity studies of lactam derivatives of MT-II and SHU-9119 their activity and selectivity at human melanocortin receptors 3, 4, and Peptides. 2007 Jun;28[6] 1191-6.