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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $23.80 | Total: $119.00 |
| 1 | 10 | $20.16 | Total: $201.60 |
| 1 | 25 | $17.08 | Total: $427.00 |
| 1 | 50 | $14.56 | Total: $728.00 |
| 1 | 100 | $12.60 | Total: $1,260.00 |
Overview
AM095 (free acid) is a potent LPA1 receptor antagonist with IC50 values of 0.98 ?M for recombinant human LPA1 and 0.73 ?M for recombinant mouse LPA1.
Chemical Properties
| Molecular Formula | C27H24N2O5 |
| Molecular Weight | 456.49 |
| CAS Numbers | 1228690-36-5 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | C[C@@H](OC(=O)Nc1c(C)noc1-c1ccc(cc1)-c1ccc(CC(O)=O)cc1)c1ccccc1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Castelino FV, et al. Amelioration of dermal fibrosis by genetic deletion or pharmacologic antagonism of lysophosphatidic acid receptor 1 in a mouse model of scleroderma. Arthritis Rheum. 2011 May;63[5] 1405-15.