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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $24.65 | Total: $123.25 |
| 1 | 10 | $20.88 | Total: $208.80 |
| 1 | 25 | $17.69 | Total: $442.25 |
| 1 | 50 | $15.08 | Total: $754.00 |
| 1 | 100 | $13.05 | Total: $1,305.00 |
Overview
L-371,257 is a competitive antagonist of oxytocin receptor with pA2 of 8.4 and Ki of 19 nM. L-371,257 shows a Ki of 3.7 nM for vasopressin receptor 1a.
Chemical Properties
| Molecular Formula | C28H33N3O6 |
| Molecular Weight | 507.58 |
| CAS Numbers | 162042-44-6 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | COc1cc(OC2CCN(CC2)C(C)=O)ccc1C(=O)N1CCC(CC1)N1C(=O)OCc2ccccc12 |
Storage and Handling
0C Short Term, -20C Long Term
References
Williams PD, et al. 1-[1-[4-[[N-acetyl-4-piperidinyl]oxy]-2-methoxybenzoyl]piperidin-4- yl]-4H-3,1-benzoxazin-2[1H]-one [L-371,257] a new, orally bioavailable, non-peptide oxytocin antagonist. J Med Chem. 1995 Nov 10;38[23] 4634-6.
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