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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $29.75 | Total: $148.75 |
| 1 | 10 | $25.20 | Total: $252.00 |
| 1 | 25 | $21.35 | Total: $533.75 |
| 1 | 50 | $18.20 | Total: $910.00 |
| 1 | 100 | $15.75 | Total: $1,575.00 |
Overview
AM095 is a potent LPA1 receptor antagonist with IC50 values of 0.98 and 0.73 ?M for recombinant human or mouse LPA1 respectively.
Chemical Properties
| Molecular Formula | C27H23N2NaO5 |
| Molecular Weight | 478.47 |
| CAS Numbers | 1345614-59-6 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | [Na+].C[C@@H](OC(=O)Nc1c(C)noc1-c1ccc(cc1)-c1ccc(CC([O-])=O)cc1)c1ccccc1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Swaney JS, et al. Pharmacokinetic and pharmacodynamic characterization of an oral lysophosphatidic acid type 1 receptor-selective antagonist. J Pharmacol Exp Ther. 2011 Mar;336[3] 693-700.