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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $26.35 | Total: $131.75 |
| 1 | 10 | $22.32 | Total: $223.20 |
| 1 | 25 | $18.91 | Total: $472.75 |
| 1 | 50 | $16.12 | Total: $806.00 |
| 1 | 100 | $13.95 | Total: $1,395.00 |
Overview
NMS-P118 is a potent, selective and orally available Inhibitor of PARP-1 for cancer therapy.
Chemical Properties
| Molecular Formula | C20H24F3N3O2 |
| Molecular Weight | 395.42 |
| CAS Numbers | 1262417-51-5 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | NC(=O)c1cc(F)cc2CN(C3CCN(CC3)C3CCC(F)(F)CC3)C(=O)c12 |
Storage and Handling
0C Short Term, -20C Long Term
References
Papeo G, et al. Discovery of 2-[1-[4,4-Difluorocyclohexyl]piperidin-4-yl]-6-fluoro-3-oxo-2,3-dihydro-1H-isoindole-4-carboxamide [NMS-P118] A Potent, Orally Available, and Highly Selective PARP-1 Inhibitor for Cancer Therapy. J Med Chem. 2015 Sep 10;58[17] 6875-98.