d[Cha4]-AVP acetate(500170-27-4 free base)

d[Cha4]-AVP acetate(500170-27-4 free base)

ATP2082L

1000 Items

$110.50

$110.50 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
15 $72.25 Total: $361.25
110 $61.20 Total: $612.00
125 $51.85 Total: $1,296.25
150 $44.20 Total: $2,210.00
1100 $38.25 Total: $3,825.00

Overview

d[Cha4]-AVP acetate is a potent and selective human vasopressin V1B receptor agonist (Ki values are 1.2, 151, 240 and 750 nM for V1B, V1A, Oxytocin and V2 receptors respectively). Stimulates ACTH and corticosterone secretion and exhibits negligible vasopressor activity in vivo.

Chemical Properties

Molecular FormulaC52H75N13O13S2
Molecular Weight1154.37
SolubilityDMSO
Purity98% by HPLC
SMILES CodeO=C(N[C@@H](CC(N)=O)C(N[C@H](C(N1CCC[C@H]1C(N[C@H](C(NCC(N)=O)=O)CCCN=C(N)N)=O)=O)CSSCCC(N[C@@H](CC2=CC=C(O)C=C2)C(N[C@@H](CC3=CC=CC=C3)C(N4)=O)=O)=O)=O)[C@@H]4CC5CCCCC5.CC(O)=O

Storage and Handling

0C Short Term, -20C Long Term

References

Derick et al [2002] [1-Deamino-4-cyclohexylalanine] arginine vasopressin a potent and specific agonist for vasopressin V1b receptors. Endocrinology 143 4655 PMID