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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $58.65 | Total: $293.25 |
| 1 | 10 | $49.68 | Total: $496.80 |
| 1 | 25 | $42.09 | Total: $1,052.25 |
| 1 | 50 | $35.88 | Total: $1,794.00 |
| 1 | 100 | $31.05 | Total: $3,105.00 |
Overview
COR659 is a 2-acylaminothiophene derivative able to suppress alcohol and chocolate self-administration in rats, likely via positive allosteric modulation of the GABAB receptor and antagonisminverse agonism at the cannabinoid CB1 receptor.
Chemical Properties
| Molecular Formula | C16H16ClNO3S |
| Molecular Weight | 337.82 |
| CAS Numbers | 544450-68-2 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CCc1c(C)sc(NC(=O)c2ccc(Cl)cc2)c1C(=O)OC |
Storage and Handling
0C Short Term, -20C Long Term
References
Francesca Ferlenghi, et al. The GABA B receptor positive allosteric modulator COR659 In vitro metabolism, in vivo pharmacokinetics in rats, synthesis and pharmacological characterization of metabolically protected derivatives. Eur J Pharm Sci. 2020 Dec 1;155 105544.