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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $72.25 | Total: $361.25 |
| 1 | 10 | $61.20 | Total: $612.00 |
| 1 | 25 | $51.85 | Total: $1,296.25 |
| 1 | 50 | $44.20 | Total: $2,210.00 |
| 1 | 100 | $38.25 | Total: $3,825.00 |
Overview
Tyrphostin AG 538 is a chalcone compound, an IGF-1 receptor kinase inhibitor (IC?0 : for 400 nM) that is potent, cell-permeable, reversible, and competitive.
Chemical Properties
| Molecular Formula | C16H11NO5 |
| Molecular Weight | 297.26 |
| CAS Numbers | 133550-18-2 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | C(C(=CC1=CC(O)=C(O)C=C1)C#N)(=O)C2=CC(O)=C(O)C=C2 |
Storage and Handling
0C Short Term, -20C Long Term
References
Blum G, et al. Substrate competitive inhibitors of IGF-1 receptor kinase. Biochemistry. 2000;39[51] 15705-15712.