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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $36.55 | Total: $182.75 |
| 1 | 10 | $30.96 | Total: $309.60 |
| 1 | 25 | $26.23 | Total: $655.75 |
| 1 | 50 | $22.36 | Total: $1,118.00 |
| 1 | 100 | $19.35 | Total: $1,935.00 |
Overview
Tyrphostin A25 (Tyrphostin AG 82) is a specific EGFR tyrosine kinase inhibitor and GPR35 agonist with an IC50 value of 0.94 ?M for GPR35 and an EC50 value of 5.3 ?M for GPR35.
Chemical Properties
| Molecular Formula | C10H6N2O3 |
| Molecular Weight | 202.17 |
| CAS Numbers | 118409-58-8 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | C(=C(C#N)C#N)C1=CC(O)=C(O)C(O)=C1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Klemke RL, et al. Receptor tyrosine kinase signaling required for integrin alpha v beta 5-directed cell motility but not adhesion on vitronectin. J Cell Biol. 1994;127[3] 859-866.