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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $43.35 | Total: $216.75 |
| 1 | 10 | $36.72 | Total: $367.20 |
| 1 | 25 | $31.11 | Total: $777.75 |
| 1 | 50 | $26.52 | Total: $1,326.00 |
| 1 | 100 | $22.95 | Total: $2,295.00 |
Overview
ASP5878 potently inhibited the tyrosine kinase activities of recombinant FGFR1, 2, 3, and 4 with IC50 values of 0.47, 0.60, 0.74, and 3.5 nmolL.
Chemical Properties
| Molecular Formula | C18H19F2N5O4 |
| Molecular Weight | 407.37 |
| CAS Numbers | 1453208-66-6 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | COc1cc(OC)c(F)c(COc2cnc(Nc3cnn(CCO)c3)nc2)c1F |
Storage and Handling
0C Short Term, -20C Long Term
References
Futami T, et al. ASP5878, a Novel Inhibitor of FGFR1, 2, 3, and 4, Inhibits the Growth of FGF19-Expressing Hepatocellular Carcinoma. Mol Cancer Ther. 2017 Jan;16[1] 68-75.