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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $24.65 | Total: $123.25 |
| 1 | 10 | $20.88 | Total: $208.80 |
| 1 | 25 | $17.69 | Total: $442.25 |
| 1 | 50 | $15.08 | Total: $754.00 |
| 1 | 100 | $13.05 | Total: $1,305.00 |
Overview
Ritanserin (R 55667) is a highly effective, relatively selective, long-acting 5-HT2 receptor antagonist (IC50: 0.9 nM), with less activity on Histamine H1, Dopamine D2, Adrenergic ?1, and Adrenergic ?2 receptors.
Chemical Properties
| Molecular Formula | C27H25F2N3OS |
| Molecular Weight | 477.57 |
| CAS Numbers | 87051-43-2 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cc1nc2sccn2c(=O)c1CCN1CCC(CC1)=C(c1ccc(F)cc1)c1ccc(F)cc1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Leysen JE, et al. Receptor-binding properties in vitro and in vivo of ritanserin A very potent and long acting serotonin-S2 antagonist. Mol Pharmacol. 1985 Jun;27[6] 600-11.