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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $81.60 | Total: $408.00 |
| 1 | 10 | $69.12 | Total: $691.20 |
| 1 | 25 | $58.56 | Total: $1,464.00 |
| 1 | 50 | $49.92 | Total: $2,496.00 |
| 1 | 100 | $43.20 | Total: $4,320.00 |
Overview
Samelisant (SUVN-G3031) is a selective and inverse agonist of H3 receptor with Kis of 8.7 nM and 9.8 nM for human and rat. Samelisant has anticataplectic effects and can be used in studies about narcolepsy.
Chemical Properties
| Molecular Formula | C21H31N3O3 |
| Molecular Weight | 373.49 |
| CAS Numbers | 1394808-82-2 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | O(C1CCN(CC1)C2CCC2)C3=CC=C(NC(CN4CCOCC4)=O)C=C3 |
Storage and Handling
0C Short Term, -20C Long Term
References
Nirogi R, et al. Samelisant [SUVN-G3031], a potent, selective and orally active histamine H3 receptor inverse agonist for the potential treatment of narcolepsy pharmacological and neurochemical characterisation. Psychopharmacology [Berl]. 2021 Jun;238[6] 1495-1511.