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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $29.75 | Total: $148.75 |
| 1 | 10 | $25.20 | Total: $252.00 |
| 1 | 25 | $21.35 | Total: $533.75 |
| 1 | 50 | $18.20 | Total: $910.00 |
| 1 | 100 | $15.75 | Total: $1,575.00 |
Overview
HIF-1 inhibitor-4 (HIF-1 inhibitor-4) is a HIF-1 inhibitor with IC50 of 560 nM. HIF-1 inhibitor-4 reduces the HIF-1? protein level without affecting its mRNA level.
Chemical Properties
| Molecular Formula | C18H19IN2O2 |
| Molecular Weight | 422.26 |
| CAS Numbers | 333357-56-5 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | IC1=CC=C(NC(=O)C2=CC=C(CN3CCOCC3)C=C2)C=C1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Nagao S, et al. Synthesis and structure-activity relationships of novel, potent, orally active hypoxia-inducible factor-1 inhibitors. Bioorg Med Chem. 2014 Oct 1;22[19] 5513-29.