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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $171.70 | Total: $858.50 |
| 1 | 10 | $145.44 | Total: $1,454.40 |
| 1 | 25 | $123.22 | Total: $3,080.50 |
| 1 | 50 | $105.04 | Total: $5,252.00 |
| 1 | 100 | $90.90 | Total: $9,090.00 |
Overview
Dual FAAHsEH-IN-1 is a dual inhibitor of sEH (soluble epoxide hydrolase) (IC50: 9.6 nM) and FAAH (fatty acid amide hydrolase) (IC50: 7 nM) with high affinity and anti-inflammatory activity.
Chemical Properties
| Molecular Formula | C25H22ClN3O3S2 |
| Molecular Weight | 512.04 |
| CAS Numbers | 2756099-59-7 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | N(C(=O)C1CCN(S(=O)(=O)C2=C(Cl)C=CC=C2)CC1)C3=CC=C(C4=NC=5C(S4)=CC=CC5)C=C3 |
Storage and Handling
0C Short Term, -20C Long Term
References
Wilt S, Kodani S, Valencia L, et al. Further exploration of the structure-activity relationship of dual soluble epoxide hydrolasefatty acid amide hydrolase inhibitors. Bioorg Med Chem. 2021;51 116507.