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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $139.40 | Total: $697.00 |
| 1 | 10 | $118.08 | Total: $1,180.80 |
| 1 | 25 | $100.04 | Total: $2,501.00 |
| 1 | 50 | $85.28 | Total: $4,264.00 |
| 1 | 100 | $73.80 | Total: $7,380.00 |
Overview
BMS-688521 BMS-688521 is an orally active and potent inhibitor of LFA-1ICAM interaction, a small molecule antagonist of leukocyte function-associated antigen-1 (LFA-1), with potential anti-inflammatory activity.
Chemical Properties
| Molecular Formula | C26H19Cl2N5O4 |
| Molecular Weight | 536.37 |
| CAS Numbers | 893397-44-9 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | O=C1[C@@]2([C@@H](CN(C2)C3=CC=C(C(O)=O)C=N3)C4=CC=C(C#N)C=C4)N(C)C(=O)N1C5=CC(Cl)=CC(Cl)=C5 |
Storage and Handling
0C Short Term, -20C Long Term
References
Watterson SH, et al. Small molecule antagonist of leukocyte function associated antigen-1 [LFA-1] structure-activity relationships leading to the identification of 6-[[5S,9R]-9-[4-cyanophenyl]-3-[3,5-dichlorophenyl]-1-methyl-2,4-dioxo-1,3,7-triazaspiro[4.4]nonan-7-yl]nicotinic acid [BMS-688521]. J Med Chem. 2010 May 13;53[9] 3814-30.