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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $22.95 | Total: $114.75 |
| 1 | 10 | $19.44 | Total: $194.40 |
| 1 | 25 | $16.47 | Total: $411.75 |
| 1 | 50 | $14.04 | Total: $702.00 |
| 1 | 100 | $12.15 | Total: $1,215.00 |
Overview
Linaprazan (AZD0865) inhibits gastric H+,K+-ATPase through K+-competitive binding, with an IC50 of 1.0 ?M.
Chemical Properties
| Molecular Formula | C21H26N4O2 |
| Molecular Weight | 366.46 |
| CAS Numbers | 248919-64-4 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cc1nc2c(NCc3c(C)cccc3C)cc(cn2c1C)C(=O)NCCO |
Storage and Handling
0C Short Term, -20C Long Term
References
Gedda K et al. Mechanism of action of AZD0865, a K+-competitive inhibitor of gastric H+,K+-ATPase. Biochem Pharmacol. 2007 Jan 15;73[2] 198-205.