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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $83.30 | Total: $416.50 |
| 1 | 10 | $70.56 | Total: $705.60 |
| 1 | 25 | $59.78 | Total: $1,494.50 |
| 1 | 50 | $50.96 | Total: $2,548.00 |
| 1 | 100 | $44.10 | Total: $4,410.00 |
Overview
H3B-120 is a highly selective, competitive, and allosteric carbamoyl phosphate synthetase 1 (CPS1) inhibitor with an IC50 of 1.5 ?M and a Ki of 1.4 ?M, exhibiting anti-cancer activity.
Chemical Properties
| Molecular Formula | C19H24N4O2S |
| Molecular Weight | 372.48 |
| CAS Numbers | 2194903-42-7 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CN(Cc1ccccc1)C(=O)N1CCC(CC1)C(=O)Nc1nc(C)cs1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Yao S, et al. Small Molecule Inhibition of CPS1 Activity through an Allosteric Pocket. Cell Chem Biol. 2020 Mar 19;27[3] 259-268.